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  • Icatibant acetate cas 138614-30-9

Hurae . 13, 2023 10:04 Hoki ki te rarangi

Icatibant acetate cas 138614-30-9



Icatibant acetate cas 138614-30-9

Ko te Icatibant Acetate he antagonist o te kaikawe bradykinin B2, ka taea te whakamahi ki te rongoa i te angioedema tuku iho.

ako in vitro

Icatibant(10-30μM)potentiatesangiotensinIII, butnotangiotensinII(contractionmediatedbyangiotensinAT1receChemicalbookptors),me Lys-des-Arg9-bradykinin,butnotdes-Arg9-bradykinin(whakaarohia e tebradykininB1receptors).

i roto i te ako vivo

Ko te Icatibant (10-30μM) te whakakaha i te angiotensin III, engari ehara i te angiotensinII(contractionmediatedbyangiotensinAT1receptors), me Lys-des-Arg9-bradykinin, butnotdes-Arg9-bradykinin(whakaarohia e tebradykininB1receptors). Tauira Kararehe:Kiore wahine o te riu CBA/J(H-Chemicalbook2k).

Inenga:0.06,0.3,1.5mg/kg ranei.

Whakahaerenga: Whakahaerenga i raro i nga wa katoa.

Hua:Ko te roanga o te inenga tino nui ko 93.6±6.8mm me te inenga 1.5mg/kg me te 94.0±4.1mm me te inenga 0.3mg/kg, e whakaatu ana i te painga aukati nui ki te poto.

Nga taonga acetate Atebant Nga tikanga rokiroki -20°C wairewa DMSO:65.0(MaxConc.mg/mL); 47.63 (MaxConc. MM) Ethanol: 0.25 (MaxConc. MgChemicalbook/mL); 0.18 (MaxConc. MM) PBS (pH7.2) : 10.0 (MaxConc. Mg/mL); 7.33(MaxConc.mM) Acrystallinesolid

nama CAS 138614-30-9

tātai rāpoi C59H89N19O13S.C2H4O2

Taumaha rāpoi 1364.59EINECS tau:-

Ko nga ahuatanga matū tinana o Altybant acetate

Kiato 1.6g/cm3

tātai rāpoi C61H93N19O15S

Te taumaha ngota 1364.57000

Papatipu tika 1363.68000

 

Icatibant acetate cas 138614-30-9

Ko te Icatibant Acetate he antagonist o te kaikawe bradykinin B2, ka taea te whakamahi ki te rongoa i te angioedema tuku iho.

  • ingoa reo Ingarihi

  • Icatibant acetate [USAN]; (R)-Arginyl-(S)-arginyl-(S)-prolyl-(2S,4R)-(4-hydroxyprolyl)glycyl-(S)-(3-(2-thienyl)alanyl)-(S)- seryl-(R)-((1,2,3,4-tetrahydro-3-isoquinolyl)carbonyl)-(2S,3aS,7aS)-((hexahydro-2-indolinyl)carbonyl)-(S)-arginine acetate (tote); Icatibant acetate; L-Arginine, D-arginyl-L-arginyl-L-prolyl-trans-4-hydroxy-L-prolylglycyl-3-(2-thienyl) -L-alanyl-L-seryl-D-1,2,3, 4-tetrahydro-3-isoquinolinecarbonyl-L-(2alpha,3abeta,7abeta)-octahydro-1H-indole-2-carbonyl-, acetate (tote)

  • ingoa ingoa Hainamana

  • Acetabant acetate; D - l-arginine base - L - arginine base - L - preserved ammonia acyl - (4 r) - 4 - hydroxy - L - preserved ammonia acyl sugar-based - 3 - (2 -) thiophene base - L - propylene ammonia acyl - L - hiraka ammonia acyl - (3 r) - 1, 2, 3, 4 - wha hauwai Puka matū - 3 - isoquinoline carbonyl - (as) 2 s, 3 rite, 7-8 h - 1 h - indole -2-carbonyl-L-arginine acetate; Aitebant acetate (Aitebant acetate, HOE140); ACETATE; Aldeibant acetate
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